4LSC2021 – PZM21

SKU: 4LSC2021 Category: Tag:

Catalog Number: 4LSC2021

CAS #: None

Name: PZM21, 1-((S)-2-(dimethylamino)-3-(4-hydroxyphenyl)propyl)-3-((S)-1-(thiophen-3-yl)propan-2-yl)urea

Product Description: Potent Gi activator with exceptional selectivity for µOR and minimal ß-arrestin-2 recruitment.

References:

Structure-based discovery of opioid analgesics with reduced side effects. Nature 1–6DOI: 10.1038/nature19112